CYCLIC PEPTIDES HAVING MELANOCORTIN-4 RECEPTOR AGONIST ACTIVITY
摘要
The presente invention refers to peptides cyclized via disulfide or lactam bridges having melanocortin-4 receptor (MC4-R) agonist activity useful for treatment of obesity.
申请公布号
CA2420058(A1)
申请公布日期
2002.03.07
申请号
CA20012420058
申请日期
2001.08.21
申请人
F. HOFFMANN-LA ROCHE AG
发明人
CHEN, LI;CHEUNG, ADRIAN WAI-HING;YAGALOFF, KEITH ALAN;WANG, YAO;SWISTOK, JOSEPH;DANHO, WALEED;CHU, XIN-JIE