发明名称 GEM-SUBSTITUTED alpha v beta 3 INTEGRIN ANTAGONISTS
摘要 The present invention relates to a class of compounds represented by Formula (I) or a pharmaceutically acceptable salt thereof, pharmaceutical compositions comprising compounds of Formula (I), and methods of selectively inhibiting or antagonizing the alpha v beta 3 and/or the alpha v beta 5 integrin.
申请公布号 WO0218340(A1) 申请公布日期 2002.03.07
申请号 WO2001US26963 申请日期 2001.08.29
申请人 PHARMACIA CORPORATION;KHANNA, ISH, KUMAR;YU, YI;FUN-LU, HWANG;CHANDRAKUMAR, NIZAL, S.;HUFF, RENEE, M.;RUSSELL, MARK, A.;BOYS, MARK, L.;SCHRETZMAN, LORI, A.;CHEN, BARBARA, B.;DESAI, BIPINCHANDRA, N.;NAGARAJAN, SRINIVASAN, RAJ;GASIECKI, ALAN, F.;PENNING, THOMAS, D.;ROGERS, THOMAS;WENDT, JOHN, ADAM;KHILEVICH, ALBERT;WANG, YAPING 发明人 KHANNA, ISH, KUMAR;YU, YI;FUN-LU, HWANG;CHANDRAKUMAR, NIZAL, S.;HUFF, RENEE, M.;RUSSELL, MARK, A.;BOYS, MARK, L.;SCHRETZMAN, LORI, A.;CHEN, BARBARA, B.;DESAI, BIPINCHANDRA, N.;NAGARAJAN, SRINIVASAN, RAJ;GASIECKI, ALAN, F.;PENNING, THOMAS, D.;ROGERS, THOMAS;WENDT, JOHN, ADAM;KHILEVICH, ALBERT;WANG, YAPING
分类号 A61K31/4375;A61K31/44;A61K31/4402;A61K31/444;A61K31/4545;A61K45/00;A61P1/02;A61P3/10;A61P3/14;A61P9/00;A61P9/10;A61P19/02;A61P19/10;A61P21/00;A61P27/02;A61P29/00;A61P31/00;A61P31/04;A61P31/10;A61P31/12;A61P35/00;A61P35/04;A61P43/00;C07D213/73;C07D213/74;C07D401/12;C07D471/04;(IPC1-7):C07D213/74;A61K31/442;A61K31/553 主分类号 A61K31/4375
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