发明名称 SUBSTITUTED 3-CYANOQUINOLINES AS PROTEIN TYROSINE KINASES INHIBITORS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
摘要 This invention provides compounds of formula (1) wherein R1, G1, G2, R4, Z, X and n are defined herein, or a pharmaceutically acceptable salt thereof, which are useful as antineoplastic agents and in the treatment of polycystic kidney disease.
申请公布号 HU0103520(A2) 申请公布日期 2002.02.28
申请号 HU20010003520 申请日期 1999.09.22
申请人 AMERICAN CYANAMID COMPANY 发明人 BERGER DAN MAARTEN;JR. FLOYD MIDDLETON BRAWNER;FROST PHILIP;HAMANN PHILIP ROSS;SALVATI MARK ERNEST;TSOU HWEI-RU;WISSNER ALLAN;ZHANG NAN
分类号 A61K31/47;A61K31/4706;A61K31/4709;A61K31/4725;A61K31/496;A61K31/502;A61K31/506;A61K31/5377;A61K31/538;A61K31/5513;A61P13/00;A61P35/00;C07D215/54;C07D215/56;C07D401/12;C07D401/14;C07D405/12;C07D405/14;C07D409/12;C07D413/12;C07D417/12;C07D417/14;C07D487/04;C07D491/04;C07D491/056;C07D491/10 主分类号 A61K31/47
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