发明名称 |
Novel guanidine mimics as factor Xa inhibitors |
摘要 |
The present application describes nitrogen containing heteroaromatics and derivatives thereof of formula I: or pharmaceutically acceptable salt forms thereof, wherein rings D-E represent guanidine mimics, which are useful as inhibitors of factor Xa.
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申请公布号 |
US2002025963(A1) |
申请公布日期 |
2002.02.28 |
申请号 |
US20010924381 |
申请日期 |
2001.08.08 |
申请人 |
LAM PATRICK Y.;CLARK CHARLES G.;DOMINGUEZ CELIA;FEVIG JOHN M.;HAN QI;LI RENHUA;PINTO DONALD JP;PRUITT JAMES R.;QUAN MIMI L. |
发明人 |
LAM PATRICK Y.;CLARK CHARLES G.;DOMINGUEZ CELIA;FEVIG JOHN M.;HAN QI;LI RENHUA;PINTO DONALD JP;PRUITT JAMES R.;QUAN MIMI L. |
分类号 |
C07D231/14;C07D231/56;C07D233/54;C07D233/61;C07D261/20;C07D401/04;C07D403/04;C07D405/04;C07D413/04;C07D413/14;(IPC1-7):C07D413/02;C0743/02;A61K31/519;A61K31/517;A61K31/470;A61K31/472;A61K31/502;A61K31/498 |
主分类号 |
C07D231/14 |
代理机构 |
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代理人 |
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地址 |
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