EFFICIENT LIGAND-MEDIATED ULLMANN COUPLING OF ANILINES AND AZOLES
摘要
The present invention provides of method of preparing phenyl-substituted azoles. This method uses an efficient ligand-accelerated Ullmann coupling reaction of anilines with azoles. The coupling products are useful for preparing factor Xa inhibitors.
申请公布号
CA2417426(A1)
申请公布日期
2002.01.31
申请号
CA20012417426
申请日期
2001.07.26
申请人
BRISTOL-MYERS SQUIBB PHARMA COMPANY
发明人
ROSSANO, LUCIUS T.;CLARK, CHARLES G.;TELEHA, CHRISTOPHER A.;LI, HUI-YIN;OH, LYNETTE M.;CONFALONE, PASQUALE N.;ZHOU, JIA CHENG