摘要 |
A method for producing (I) or (II), characterized in that (III) and (IV) are reacted (1) in a secondary or tertiary alcohol in the presence of a base or (2) in the absence of a base. The method can be employed for producing a 1-substituted-1,2,3-triazole compound having inhibitory action for tyrosine kinase, in a high yield and with a simple and easy process, on a commercial scale.
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申请人 |
TAKEDA CHEMICAL INDUSTRIES, LTD.;IKEMOTO, TOMOMI;ITO, TATSUYA;TOMIMATSU, KIMINORI;SAWAI, YASUHIRO;NISHIYAMA, HIROHIKO;ISOGAMI, YASUSHI |
发明人 |
IKEMOTO, TOMOMI;ITO, TATSUYA;TOMIMATSU, KIMINORI;SAWAI, YASUHIRO;NISHIYAMA, HIROHIKO;ISOGAMI, YASUSHI |