发明名称 METHOD FOR PRODUCING 1-SUBSTITUTED-1,2,3-TRIAZOLE DERIVATIVE
摘要 A method for producing (I) or (II), characterized in that (III) and (IV) are reacted (1) in a secondary or tertiary alcohol in the presence of a base or (2) in the absence of a base. The method can be employed for producing a 1-substituted-1,2,3-triazole compound having inhibitory action for tyrosine kinase, in a high yield and with a simple and easy process, on a commercial scale.
申请公布号 WO0206249(A1) 申请公布日期 2002.01.24
申请号 WO2001JP06145 申请日期 2001.07.16
申请人 TAKEDA CHEMICAL INDUSTRIES, LTD.;IKEMOTO, TOMOMI;ITO, TATSUYA;TOMIMATSU, KIMINORI;SAWAI, YASUHIRO;NISHIYAMA, HIROHIKO;ISOGAMI, YASUSHI 发明人 IKEMOTO, TOMOMI;ITO, TATSUYA;TOMIMATSU, KIMINORI;SAWAI, YASUHIRO;NISHIYAMA, HIROHIKO;ISOGAMI, YASUSHI
分类号 A61P9/10;A61P31/12;A61P31/18;A61P35/00;A61P43/00;C07D249/04;(IPC1-7):C07D249/04;C07D413/12;C07D263/32;A61K31/422 主分类号 A61P9/10
代理机构 代理人
主权项
地址
您可能感兴趣的专利