发明名称 |
METHOD FOR SYNTHESIS OF HALOPYRIDYL-ACYCLOPENTANE DERIVATIVE AND INTERMEDIATE THEREOF |
摘要 |
The present invention relates to a method for synthesis of an optically active halopyridyl-azacyclo-pentane derivative and the intermediate thereof which comprises preparing an optically active allene-1,3-dicarboxylic acid ester derivative from an optically active acetonedicarboxylic acid ester derivative and then proceeding through a 7-azabicyclo[2.2.1]heptane derivative to obtain the objective product.
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申请公布号 |
US2002010339(A1) |
申请公布日期 |
2002.01.24 |
申请号 |
US20000462379 |
申请日期 |
2000.01.07 |
申请人 |
NODE MANABU;NAKAMURA DAISAKU;FUJIWARA TOSHIO;ICHIHASHI SHOGO |
发明人 |
NODE MANABU;NAKAMURA DAISAKU;FUJIWARA TOSHIO;ICHIHASHI SHOGO |
分类号 |
C07D487/04;(IPC1-7):A61K9/00;C07D213/54;C07D213/53;C07D213/36;C07D213/26;C07D211/82;C07D211/70 |
主分类号 |
C07D487/04 |
代理机构 |
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主权项 |
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地址 |
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