发明名称 |
1-(6-Methylpyridin-3-yl)-2-[(4-(methylsulfonyl)phenyl]ethanone and process for preparing thereof |
摘要 |
<p>1-(6-Methylpyridin-3-yl)-2-(4-methylsulfonyl-phenyl)-ethanone is new. 1-(6-methylpyridin-3-yl)-2-(4-methylsulfonyl-phenyl)-ethanone of formula (I) is new: Independent claims are also included for the following: (a) a 4-step preparation of (I) where the third step for the preparation of N,N-dialkylamino-(6-methyl-3-pyridyl)acetonitriles of formula (III) and the last step are claimed per se; (b) compounds (III); (c) alkali metal 1-hydroxy-(6-methylpyridin-3-yl)methanesulfonate intermediates of formula (II) (for preparing (III)); (d) preparation of (II) comprising treating 2-methyl-5-vinylpyridine with ozone followed by reduction with an alkali hydrogen sulfite. R1, R2 = 1-4C alkyl; M = alkali metal.</p> |
申请公布号 |
CZ20012457(A3) |
申请公布日期 |
2002.01.16 |
申请号 |
CZ20010002457 |
申请日期 |
2000.01.13 |
申请人 |
LONZA AG;MERCK & CO., INC. |
发明人 |
ARMBRUSTER ERICH;BESSARD YVES;KUO DAVID;LERESCHE JAMES EDWARD;PROPLESCH RALF;RODUIT JEAN-PAUL |
分类号 |
C07D213/50;C07D213/52;C07D213/53;C07D213/57;(IPC1-7):C07D213/50 |
主分类号 |
C07D213/50 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|