发明名称 CYCLOPENTYL-SUBSTITUTED GLUTARAMIDE DERIVATIVES AS INHIBITORS OF NEUTRAL ENDOPEPTIDASE
摘要 The invention provides compounds of formula I wherein R1 is optionally substituted C1-6alkyl, optionally substituted C3-7 cycloalkyl, optionally substituted aryl or optionally substituted heterocyclyl; n is 0, 1 or 2; and Y is -NR18S(O)uR19 or a group shown below.
申请公布号 CA2414881(A1) 申请公布日期 2002.01.10
申请号 CA20012414881 申请日期 2001.07.02
申请人 PFIZER INC. 发明人 MAW, GRAHAM NIGEL;COOK, ANDREW SIMON;BARBER, CHRISTOPHER GORDON;STOBIE, ALAN;PRYDE, DAVID CAMERON
分类号 A61K;A61K31/00;A61K31/19;A61K31/195;A61K31/196;A61K31/343;A61K31/36;A61K31/40;A61K31/4015;A61K31/4045;A61K31/433;A61K31/4402;A61K31/4406;A61K31/4412;A61K31/4453;A61K31/45;A61K31/495;A61K31/535;A61K45/06;A61P;A61P15/00;A61P43/00;C07C;C07C233/58;C07C233/60;C07C235/40;C07C237/22;C07C237/24;C07C275/52;C07C311/13;C07C311/18;C07C311/51;C07D;C07D207/14;C07D207/26;C07D207/27;C07D209/14;C07D211/40;C07D211/76;C07D213/64;C07D213/70;C07D213/71;C07D213/74;C07D213/75;C07D285/12;C07D285/135;C07D307/81;C07D317/58;(IPC1-7):C07C237/22;C07D209/16 主分类号 A61K
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