发明名称 DERIVATIVES OF QUINOLINE AS ALPHA-2 ANTAGONISTS
摘要 The invention provides a compound of formula (I), wherein A, Ra, Rb, R1 to R5, m and t are as defined as disclosed, or a pharmaceutically acceptable salt or ester thereof, useful as alpha-2 antagonist. The compounds I can be used for the treatment of diseases or conditions wherein alpha-2 antagonists are indicated to be effective.
申请公布号 WO0164645(A3) 申请公布日期 2001.12.27
申请号 WO2001FI00203 申请日期 2001.02.28
申请人 ORION CORPORATION;OY JUVANTIA PHARMA LTD;WURSTER, SIEGFRIED;ENGSTROEM, MIA;SAVOLA, JUHA-MATTI;HOEGLUND, IISA;SALLINEN, JUKKA;HAAPALINNA, ANTTI;TAUBER, ANDREI;HOFFREN, ANNA-MARJA;SALO, HARRI 发明人 WURSTER, SIEGFRIED;ENGSTROEM, MIA;SAVOLA, JUHA-MATTI;HOEGLUND, IISA;SALLINEN, JUKKA;HAAPALINNA, ANTTI;TAUBER, ANDREI;HOFFREN, ANNA-MARJA;SALO, HARRI
分类号 C07D215/46;A61K31/4709;A61K31/473;A61K31/4748;A61K31/496;A61K31/5377;A61P3/04;A61P3/10;A61P9/02;A61P15/10;A61P25/00;A61P25/02;A61P25/16;A61P25/18;A61P25/22;A61P25/24;A61P25/28;A61P43/00;C07D215/00;C07D215/44;C07D215/48;C07D219/10;C07D221/16;C07D221/22;C07D401/12;(IPC1-7):C07D215/44;C07D221/04;C07D221/06;C07D221/18;C07D241/04;A61K31/470;A61K31/474 主分类号 C07D215/46
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