发明名称 NOVEL SUBSTITUTED PYRAZOLO[4,3-<i>e</i>]DIAZEPINES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, USE AS MEDICINAL PRODUCTS AND PROCESSES FOR PREPARING THEM
摘要 The invention relates to novel substituted pyrazolo[4,3-e]- diazepines of general formula (I), to pharmaceutical compositions containing them, to their use as medicinal products and to processes for preparing them. The compounds are selective PDE4 inhibitors.
申请公布号 WO0149689(A3) 申请公布日期 2001.12.20
申请号 WO2000EP13380 申请日期 2000.12.27
申请人 WARNER-LAMBERT COMPANY;BURNOUF, CATHERINE;BERECIBAR, AMAYA;NAVET, MICHEL 发明人 BURNOUF, CATHERINE;BERECIBAR, AMAYA;NAVET, MICHEL
分类号 A61K31/5517;A61P1/00;A61P7/00;A61P9/04;A61P9/08;A61P9/12;A61P11/00;A61P11/06;A61P17/00;A61P17/02;A61P17/06;A61P19/02;A61P19/10;A61P25/00;A61P25/22;A61P25/24;A61P29/00;A61P31/18;A61P35/00;A61P37/02;A61P37/08;A61P43/00;C07D487/04;(IPC1-7):C07D487/04;A61K31/551 主分类号 A61K31/5517
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