发明名称 PROCESS FOR THE SYNTHESIS OF (2R, 2-ALPHA-R, 3A)-2-[1-(3,5-BIS(TRIFLUOROMETHYL)PHENYL)ETHOXY]-3-(4-FLUOROPHENYL)-1,4-OXAZINE
摘要 The present invention is concerned with novel processes for the preparation of (2R, 2-alpha-R, 3a)-2-[1-[3,5-bis(trifluoromethyl)phenyl]ethoxy-3-(4-fluorophenyl)-1,4-oxazine. This compound is useful as an intermediate in the synthesis of compounds which possess pharmacological activity.
申请公布号 WO0194324(A1) 申请公布日期 2001.12.13
申请号 WO2001US18042 申请日期 2001.06.04
申请人 MERCK & CO., INC.;BRANDS, KAREL, M., JOS;TSAY, FUH-RONG;CONRAD, KAREN, M.;ZHAO, MATTHEW, M. 发明人 BRANDS, KAREL, M., JOS;TSAY, FUH-RONG;CONRAD, KAREN, M.;ZHAO, MATTHEW, M.
分类号 C07B61/00;C07D265/32;(IPC1-7):C07D265/32 主分类号 C07B61/00
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