发明名称 Process for Cis-1-{2-[4-(6-methoxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl)phenoxy]ethyl}pyrrolidine
摘要 This invention provides an improved process for cis-1-{2-[4-(6-methoxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl)phenoxy]ethyl}pyrrolidine which is an intermediate for the preparation of (-)cis-6-phenyl-5-[4-(2-pyrrolidin-1-yl-ethoxy)-phenyl]-5,6,7,8-tetrahydronaphthalene-2-ol which is useful for the treatment of osteoporosis.
申请公布号 US6323345(B1) 申请公布日期 2001.11.27
申请号 US20010794382 申请日期 2001.02.27
申请人 PFIZER INC. 发明人 CHIU CHARLES K. F.
分类号 C07D295/08;A61P19/10;C07C43/20;C07C43/21;C07C43/215;C07C45/48;C07C45/59;C07C49/84;C07D207/08;C07D207/34;C07D295/092;C07D317/18;C07D317/22;C07D317/26;(IPC1-7):C07D207/04 主分类号 C07D295/08
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