Inhibitors of trypsin-like enzymes

摘要

Pharmaceutical compositions comprising compounds of the formula:in which X=H or is an N-protecting group; Y is 1-10 á-amino acids; Q1 and Q2 taken together represent the residue of a diol; R is C1-4alkyl; and the asymmetric carbon atom marked * may have the D- or L-configuration, are useful in therapeutic methods of inhibiting thrombin.