发明名称 |
NOVEL PROCESS FOR PRODUCING FUSED IMIDAZOPYRIDINE DERIVATIVE AND NOVEL CRYSTAL FORM |
摘要 |
A process for producing a compound represented by the formula (I) (wherein R is an aromatic heterocycle, etc. and A is a heteroalicyclic group, etc.), characterized by reacting a compound represented by the formula (II) (wherein Hal is halogeno, and R and A have the same meanings as the above) in the presence of a sulfinic acid salt and a salt of an acid or organic base; and a novel crystal of 2-(3-isooxazolyl)-3,6,7,9-tetrahydroimidazo[4,5-d]pyrano[4,3-b]pyridine phosphate monohydrate.
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申请公布号 |
WO0174821(A1) |
申请公布日期 |
2001.10.11 |
申请号 |
WO2001JP02620 |
申请日期 |
2001.03.29 |
申请人 |
SHIONOGI & CO., LTD.;MATSUBARA, FUMIHIKO;OHYA, TAKASHI;UENAKA, MASAAKI |
发明人 |
MATSUBARA, FUMIHIKO;OHYA, TAKASHI;UENAKA, MASAAKI |
分类号 |
C07D487/04;C07D491/02;C07D491/14;C07D491/147;(IPC1-7):C07D491/147 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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