发明名称 Method of preparing alkylated salicylamides via a dicarboxylate intermediate
摘要 The present invention relates to a method of preparing an alkylated salicylamide from a protected and activated salicylamide via a dicarboxylated salicylamide intermediate. The present invention also relates to dicarboxylic salicylamide delivery agent compounds for the delivery of active agents. Methods of administration are provided as well.
申请公布号 AU8148301(A) 申请公布日期 2001.10.03
申请号 AU20010081483 申请日期 2001.03.21
申请人 EMISPHERE TECHNOLOGIES, INC. 发明人 JOSEPH N. BERNADINO;DORIS C. O'TOOLE;WILLIAM E. BAY
分类号 C07D265/36;A61K45/00;A61K47/16;A61P1/04;A61P3/00;A61P3/02;A61P5/06;A61P7/00;A61P7/02;A61P9/00;A61P9/08;A61P9/12;A61P11/06;A61P13/00;A61P15/00;A61P19/08;A61P19/10;A61P31/00;A61P35/00;A61P37/02;A61P37/08;A61P43/00;C07C231/12;C07C235/60;C07C269/00;C07C271/64;C07D265/22;C07D265/26 主分类号 C07D265/36
代理机构 代理人
主权项
地址