发明名称 METHOD OF PREPARING ALKYLATED SALICYLAMIDES VIA A DICARBOXYLATE INTERMEDIATE
摘要 <p>The present invention relates to a method of preparing an alkylated salicylamide from a protected and activated salicylamide via a dicarboxylated salicylamide intermediate. The present invention also relates to dicarboxylic salicylamide delivery agent compounds for the delivery of active agents. Methods of administration are provided as well.</p>
申请公布号 WO0170219(A1) 申请公布日期 2001.09.27
申请号 WO2001US09154 申请日期 2001.03.21
申请人 EMISPHERE TECHNOLOGIES, INC.;BERNADINO, JOSEPH, N.;O'TOOLE, DORIS, C.;BAY, WILLIAM, E. 发明人 BERNADINO, JOSEPH, N.;O'TOOLE, DORIS, C.;BAY, WILLIAM, E.
分类号 C07D265/36;A61K45/00;A61K47/16;A61P1/04;A61P3/00;A61P3/02;A61P5/06;A61P7/00;A61P7/02;A61P9/00;A61P9/08;A61P9/12;A61P11/06;A61P13/00;A61P15/00;A61P19/08;A61P19/10;A61P31/00;A61P35/00;A61P37/02;A61P37/08;A61P43/00;C07C231/12;C07C235/60;C07C269/00;C07C271/64;C07D265/22;C07D265/26;(IPC1-7):A61K31/195;C07C237/00;C07C233/00;C07C229/00;C07D265/12;C07C235/00;C07C239/00 主分类号 C07D265/36
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