METHOD OF PREPARING ALKYLATED SALICYLAMIDES VIA A DICARBOXYLATE INTERMEDIATE
摘要
<p>The present invention relates to a method of preparing an alkylated salicylamide from a protected and activated salicylamide via a dicarboxylated salicylamide intermediate. The present invention also relates to dicarboxylic salicylamide delivery agent compounds for the delivery of active agents. Methods of administration are provided as well.</p>
申请公布号
WO0170219(A1)
申请公布日期
2001.09.27
申请号
WO2001US09154
申请日期
2001.03.21
申请人
EMISPHERE TECHNOLOGIES, INC.;BERNADINO, JOSEPH, N.;O'TOOLE, DORIS, C.;BAY, WILLIAM, E.
发明人
BERNADINO, JOSEPH, N.;O'TOOLE, DORIS, C.;BAY, WILLIAM, E.