发明名称 Prevention of loss and restoration of bone mass by certain prostaglandin agonists
摘要 Prostaglandin agonists of formula (I), in which, for example, A is a sulphonyl or acyl group, B is N or CH, M contains a ring and K and Q are linking groups, methods of using such prostaglandin agonists, pharmaceutical compositions containing such prostaglandin agonists and kits useful for the treatment of bone disorders including osteoporosis.
申请公布号 US6288120(B1) 申请公布日期 2001.09.11
申请号 US19990331081 申请日期 1999.06.11
申请人 PFIZER INC. 发明人 CAMERON KIMBERLY O.;KE HUA Z.;LEFKER BRUCE A.;ROSATI ROBERT L.;THOMPSON DAVID D.
分类号 C07D249/08;A61K31/16;A61K31/18;A61K31/192;A61K31/195;A61K31/197;A61K31/341;A61K31/343;A61K31/357;A61K31/36;A61K31/381;A61K31/4015;A61K31/41;A61K31/4192;A61K31/4245;A61K31/426;A61K31/4402;A61K31/4406;A61K31/4535;A61K31/47;A61K31/4709;A61K31/4965;A61K31/505;A61K31/557;A61K33/16;A61K38/04;A61K38/22;A61K38/27;A61K45/00;A61K45/06;A61P1/02;A61P13/12;A61P19/08;A61P19/10;A61P43/00;C07C233/47;C07C235/34;C07C311/04;C07C311/06;C07C317/44;C07C323/25;C07C323/49;C07C323/59;C07D207/26;C07D207/263;C07D207/27;C07D209/14;C07D213/34;C07D213/42;C07D215/18;C07D239/26;C07D241/12;C07D249/06;C07D257/04;C07D271/12;C07D277/20;C07D277/28;C07D277/56;C07D307/24;C07D307/52;C07D307/68;C07D307/81;C07D317/58;C07D319/18;C07D333/18;C07D333/20;C07D333/24;C07D333/34;C07D333/38;C07D333/40;C07D333/58;C07D409/12;(IPC1-7):A61K31/16;A61K31/19;C07C303/00;C07C59/48 主分类号 C07D249/08
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