发明名称 FAP-ACTIVATED ANTI-TUMOR COMPOUNDS
摘要 The invention relates to a prodrug that is capable of being converted into a drug by the catalytic action of human fibroblast activation protein (FAP alpha ), said prodrug having a cleavage site which is recognised by FAP alpha , and said drug being cytotoxic or cytostatic under physiological conditions.
申请公布号 WO0071571(A3) 申请公布日期 2001.09.07
申请号 WO2000EP04261 申请日期 2000.05.11
申请人 BOEHRINGER INGELHEIM;PARK, JOHN, EDWARD;RETTIG, WOLFGANG, J.;LENTER, MARTIN;PETERS, STEFAN;MACK, JUERGEN;LEIPERT, DIETMAR;GARIN-CHESA, PILAR;FIRESTONE, RAYMOND, ARMAND;TELAN, LEILA, A. 发明人 PARK, JOHN, EDWARD;RETTIG, WOLFGANG, J.;LENTER, MARTIN;PETERS, STEFAN;MACK, JUERGEN;LEIPERT, DIETMAR;GARIN-CHESA, PILAR;FIRESTONE, RAYMOND, ARMAND;TELAN, LEILA, A.
分类号 A61K31/704;A61K38/00;A61K45/00;A61K47/42;A61K47/48;A61P35/00;A61P43/00;C07H15/252;C07K1/06;C07K1/107;C07K5/06;C07K5/062;C07K5/11;C07K5/117;(IPC1-7):C07K1/107;C07K9/00;A61K38/04 主分类号 A61K31/704
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