发明名称 |
DERIVATIVES OF QUINOLINE AS ALPHA-2 ANTAGONISTS |
摘要 |
The invention provides a compound of formula (I), wherein A, Ra, Rb, R1 to R 5, m and t are as defined as disclosed, or a pharmaceutically acceptable salt o r ester thereof, useful as alpha-2 antagonist. The compounds I can be used for the treatment of diseases or conditions wherein alpha-2 antagonists are indicated to be effective.
|
申请公布号 |
CA2400657(A1) |
申请公布日期 |
2001.09.07 |
申请号 |
CA20012400657 |
申请日期 |
2001.02.28 |
申请人 |
ORION CORPORATION;OY JUVANTIA PHARMA LTD. |
发明人 |
SAVOLA, JUHA-MATTI;SALO, HARRI;HOGLUNG, IISA;HOFFREN, ANNA-MARJA;TAUBER, ANDREI;ENGSTROM, MIA;SALLINEN, JUKKA;WURSTER, SIEGFRIED;HAAPALINNA, ANTTI |
分类号 |
C07D215/46;A61K31/4709;A61K31/473;A61K31/4748;A61K31/496;A61K31/5377;A61P3/04;A61P3/10;A61P9/02;A61P15/10;A61P25/00;A61P25/02;A61P25/16;A61P25/18;A61P25/22;A61P25/24;A61P25/28;A61P43/00;C07D215/00;C07D215/44;C07D215/48;C07D219/10;C07D221/16;C07D221/22;C07D401/12;(IPC1-7):C07D215/44;C07D221/04;C07D241/04;C07D221/06;C07D221/18;A61K31/470;A61K31/474 |
主分类号 |
C07D215/46 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|