发明名称 |
BUPROPION METABOLITES AND METHODS OF THEIR SYNTHESIS AND USE |
摘要 |
Methods and compositions are disclosed which utilize metabolites of bupropion for treating disorders ameliorated by inhibition of neuronal monoamine reuptake. Such disorders include, but are not limited to, sexual dysfunction, affective disorders, cerebral function disorders, cigarette smoking, and incontinence. Methods of making optically pure bupropion metabolites are also disclosed.
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申请公布号 |
WO0162257(A2) |
申请公布日期 |
2001.08.30 |
申请号 |
WO2000US23080 |
申请日期 |
2000.08.23 |
申请人 |
SEPRACOR INC. |
发明人 |
FANG, QUN, K.;SENANAYAKE, CHRISANTHA, H.;GROVER, PAUL |
分类号 |
A61K31/133;A61K9/08;A61K9/10;A61K9/70;A61K31/00;A61K31/135;A61K31/137;A61K31/165;A61K31/415;A61K31/4178;A61K31/43;A61K31/435;A61K31/4375;A61K31/439;A61K31/4427;A61K31/46;A61K31/465;A61K31/50;A61K31/53;A61K31/535;A61K31/537;A61K31/5375;A61K45/00;A61K45/06;A61P1/08;A61P13/00;A61P13/10;A61P15/10;A61P25/00;A61P25/08;A61P25/16;A61P25/20;A61P25/24;A61P25/28;A61P25/34;A61P43/00;C07B57/00;C07C45/51;C07C45/63;C07C49/76;C07C49/807;C07C49/82;C07C49/84;C07C213/00;C07C215/30;C07C225/16;C07C317/14;C07D265/32;(IPC1-7):A61K31/537 |
主分类号 |
A61K31/133 |
代理机构 |
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代理人 |
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地址 |
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