发明名称 Substituted oxoazaheterocyclyl compounds.
摘要 <p>This invention is directed to oxoazaheterocyclyl compounds which inhibit Factor Xa, to oxoazaheterocyclyl compounds which inhibit both Factor Xa and Factor IIa, to pharmaceutical compositions comprising these compounds, to intermediates useful for preparing these compounds, to a method of directly inhibiting Factor Xa and to a method of simultaneously directly inhibiting Factor Xa and Factor IIa.</p>
申请公布号 WO0107436(A3) 申请公布日期 2001.08.23
申请号 WO2000IB01156 申请日期 2000.07.26
申请人 AVENTIS PHARMACEUTICALS PRODUCTS INC.;EWING, WILLIAM, R.;BECKER, MICHAEL, R.;CHOI-SLEDESKI, YONG, MI.;PAULS, HEINZ, W.;HE, WEI;CONDON, STEPHEN, M;DAVIS, RODERICK, S.;HANNEY BARBARA A;SPADA, ALFRED, P.;BURNS, CHRISTOPHER, J.;JIANG, JOHN, Z.;LI, AIWEN;MYERS, MICHAEL, R.;LAU, WAN, F.;POLI, GREGORY, B. 发明人 EWING, WILLIAM, R.;BECKER, MICHAEL, R.;CHOI-SLEDESKI, YONG MI;PAULS, HEINZ, W.;HE, WEI;CONDON, STEPHEN, M.;DAVIS, RODERICK, S.;HANNEY, BARBARA, A.;SPADA, ALFRED, P.;BURNS, CHRISTOPHER, J.;JIANG, JOHN, Z.;LI, AIWEN;MYERS, MICHAEL, R.;LAU, WAN, F.;POLI, GREGORY, B.
分类号 C07D241/08;A61K31/495;A61K31/496;A61K31/498;A61K31/502;A61K31/506;A61K31/517;A61K31/519;A61K31/5377;A61P7/02;A61P9/02;A61P9/04;A61P9/10;A61P19/02;A61P25/28;A61P35/00;A61P41/00;A61P43/00;C07D401/06;C07D401/14;C07D403/06;C07D403/14;C07D405/14;C07D409/06;C07D409/12;C07D409/14;C07D413/14;C07D417/14;C07D471/04;C07D495/04;(IPC1-7):C07D403/06;C07D491/04 主分类号 C07D241/08
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