发明名称 SERINE PROTEASE INHIBITORS
摘要 Compounds having structure (A) are useful to inhibit serine protease enzymes, such as TF/factor VIIa, factor Xa, thrombin and kallikrein. These compounds may be used in methods of preventing and/or treating clotting disorders.
申请公布号 WO0041531(A3) 申请公布日期 2001.08.16
申请号 WO2000US00673 申请日期 2000.01.11
申请人 GENENTECH, INC.;ALIAGAS-MARTIN, IGNACIO;ARTIS, DEAN, R.;DINA, MICHAEL, S.;FLYGARE, JOHN, A.;GOLDSMITH, RICHARD, A.;MUNROE, REGINA, A.;OLIVERO, ALAN, G.;PASTOR, RICHARD;RAWSON, THOMAS, E.;ROBARGE, KIRK, D.;SUTHERLIN, DANIEL, P.;WEESE, KENNETH, J.;ZHOU, AIHE;ZHU, YAN 发明人 ALIAGAS-MARTIN, IGNACIO;ARTIS, DEAN, R.;DINA, MICHAEL, S.;FLYGARE, JOHN, A.;GOLDSMITH, RICHARD, A.;MUNROE, REGINA, A.;OLIVERO, ALAN, G.;PASTOR, RICHARD;RAWSON, THOMAS, E.;ROBARGE, KIRK, D.;SUTHERLIN, DANIEL, P.;WEESE, KENNETH, J.;ZHOU, AIHE;ZHU, YAN
分类号 C07D333/34;A61K31/18;A61K31/196;A61K31/216;A61K31/381;A61P7/02;A61P9/10;C07C257/18;C07C311/05;C07C311/08;C07C311/13;C07C311/18;C07C311/29;C07C311/51;(IPC1-7):C07C311/51;C07C311/06;C07C311/21;C07C257/16 主分类号 C07D333/34
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