发明名称 (HETERO)BICYCLYMETHANESULFONYLAMINO-SUBSTITUTED HYDROXAMIC ACID DERIVATIVES
摘要 Compounds of formula (I) wherein R is hydrogen, alkyl, alkenyl, alkynyl, aryl, heteroaryl or heterocyclyl; and R<1> is bicyclyl or heterobicyclyl; are useful in the treatment and prophylaxis of conditions mediated by s-CD23 or TNF.
申请公布号 WO0147874(A1) 申请公布日期 2001.07.05
申请号 WO2000GB04941 申请日期 2000.12.21
申请人 SMITHKLINE BEECHAM P.L.C.;BRUTON, GORDON;FALLER, ANDREW;ORLEK, BARRY, SIDNEY;RANA, KISHORE, K.;WALKER, GRAHAM 发明人 BRUTON, GORDON;FALLER, ANDREW;ORLEK, BARRY, SIDNEY;RANA, KISHORE, K.;WALKER, GRAHAM
分类号 C07D333/16;A61K31/18;A61K31/381;A61K31/4035;A61K31/405;A61K31/4155;A61K31/5377;A61P1/14;A61P7/00;A61P7/04;A61P9/10;A61P23/00;A61P25/00;A61P25/28;A61P29/00;A61P29/02;A61P31/00;A61P37/02;A61P37/06;A61P37/08;A61P43/00;C07C303/12;C07C303/40;C07C311/13;C07C311/19;C07D209/20;C07D209/24;C07D333/24;C07D333/52;C07D333/54;C07D333/60;C07D333/62;C07D409/12;C07D521/00;(IPC1-7):C07C311/13;C07D209/18;C07D295/185;A61K31/38;A61K31/40;A61K31/537 主分类号 C07D333/16
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