发明名称 Proliposome powders for inhalation stabilised by racemic alpha-tocopherol
摘要 The proliposome powder comprises discrete particles each comprising in a single phase; (1) a biologically active component selected from antiinflammatory and bronchorelaxing drugs, antihistamines, cyclooxygenase inhibitors, leukotriene synthesis inhibitors, leukotriene antagonists, phospholipase-A2 inhibitors, platelet aggregating factor antagonists, antiarrhythmic drugs, tranquilisers, cardiac glycosides, hormones, anti-hypertensive drugs, antidiabetic, antiparisitic and anticancer drugs, sedatives, analgesic drugs, antibiotics, antirheumatic drugs, immunotherapies, antifungal drugs, antihypotension drugs, vaccines, antiviral drugs, proteins, peptides and vitamins; (2) a stabilising proportion of tocopherol; and (3) a lipid or mixture of lipids having a phase transition temperature of below 37°C.
申请公布号 NZ501672(A) 申请公布日期 2001.06.29
申请号 NZ19980501672 申请日期 1998.06.08
申请人 ASTRA AKTIEBOLAG 发明人 NILSSON, PER-GUNNAR;BYSTROM, KATARINA
分类号 A61K9/00;A61K9/127;A61K9/72;A61K31/56;A61K47/22;(IPC1-7):A61K9/127 主分类号 A61K9/00
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