发明名称 NON PEPTIDE TACHYKININ RECEPTOR ANTAGONISTS
摘要 Compounds of Formula (I) are specific tachykinin receptor antagonists where R, m, X, R1, R2, n, Y, R3, R4, R5, and R6 are as described in the specification. The compounds are useful agents for treating conditions associated with aberrant neovascularization such as rheumatoid arthritis, atherosclerosis and tumour cell growth.
申请公布号 WO0146176(A2) 申请公布日期 2001.06.28
申请号 WO2000EP13349 申请日期 2000.12.21
申请人 WARNER-LAMBERT COMPANY;HORWELL, DAVID, CHRISTOPHER;LEWTHWAITE, RUSSELL, ANDREW;PRITCHARD, MARTIN, CLIVE;RAPHY, JENNIFER;BARTH, HUBERT;STEINER, KLAUS;SCHIEFERMAYR, BERND 发明人 HORWELL, DAVID, CHRISTOPHER;LEWTHWAITE, RUSSELL, ANDREW;PRITCHARD, MARTIN, CLIVE;RAPHY, JENNIFER;BARTH, HUBERT;STEINER, KLAUS;SCHIEFERMAYR, BERND
分类号 A61K31/404;A61K51/00;A61P1/00;A61P1/04;A61P1/08;A61P3/04;A61P9/10;A61P11/00;A61P11/02;A61P11/04;A61P11/06;A61P15/10;A61P17/00;A61P17/06;A61P19/02;A61P25/00;A61P25/04;A61P25/06;A61P25/14;A61P25/18;A61P25/22;A61P25/28;A61P29/00;A61P35/00;A61P37/08;A61P43/00;C07D405/12;(IPC1-7):C07D405/12;C07D209/20;A61K31/405;A61K31/343 主分类号 A61K31/404
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