发明名称 SACCHARIN DERIVATIVES AS ORALLY ACTIVE ELASTASE INHIBITORS
摘要 Orally active compounds of general formula (I) wherein R<1> is methyl, ethyl or 2-morpholino-ethyl group, R<2> is piperidino, morpholino or 4-methyl-piperazinyl group, n is 2 or 3 and their salts, solvates and hydrates.
申请公布号 WO0144245(A1) 申请公布日期 2001.06.21
申请号 WO2000HU00130 申请日期 2000.12.14
申请人 SANOFI-SYNTHELABO;ARANYI, PETER;BATORI, SANDOR;DESSILLA, STEPHANE;HERMECZ, ISTVAN;KAPUI, ZOLTAN;LEVAI, FERENC;MIKUS, ENDRE;PASCAL, MARC;T. NAGY, LAJOS;SIMONOT, BRUNO;URBAN SZABO, KATALIN;VARGA, MARTON;VASVARINE DEBRECZY, LELLE 发明人 ARANYI, PETER;BATORI, SANDOR;DESSILLA, STEPHANE;HERMECZ, ISTVAN;KAPUI, ZOLTAN;LEVAI, FERENC;MIKUS, ENDRE;PASCAL, MARC;T. NAGY, LAJOS;SIMONOT, BRUNO;URBAN SZABO, KATALIN;VARGA, MARTON;VASVARINE DEBRECZY, LELLE
分类号 A61K31/519;A61K31/5377;A61P1/04;A61P1/16;A61P1/18;A61P9/10;A61P9/12;A61P11/00;A61P11/06;A61P13/10;A61P13/12;A61P17/00;A61P17/02;A61P17/06;A61P19/06;A61P25/00;A61P27/16;A61P29/00;A61P31/04;A61P31/10;A61P33/02;A61P33/12;A61P35/00;A61P37/02;A61P43/00;C07D471/04;(IPC1-7):C07D471/04;A61K31/505 主分类号 A61K31/519
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