SACCHARIN DERIVATIVES AS ORALLY ACTIVE ELASTASE INHIBITORS
摘要
Orally active compounds of general formula (I) wherein R1 is methyl, ethyl o r 2-morpholino-ethyl group, R2 is piperidino, morpholino or 4-methyl-piperazin yl group, n is 2 or 3 and their salts, solvates and hydrates.
申请公布号
CA2395486(A1)
申请公布日期
2001.06.21
申请号
CA20002395486
申请日期
2000.12.14
申请人
SANOFI-SYNTHELABO
发明人
VASVARINE DEBRECZY, LELLE;ARANYI, PETER;BATORI, SANDOR;DESSILLA, STEPHANE;HERMECZ, ISTVAN;T. NAGY, LAJOS;PASCAL, MARC;MIKUS, ENDRE;KAPUI, ZOLTAN;LEVAI, FERENC;VARGA, MARTON;SIMONOT, BRUNO;URBAN SZABO, KATALIN