发明名称 TRICYCLIC INHIBITORS OF POLY(ADP-RIBOSE) POLYMERASES
摘要 Compounds of the formula (I) are poly(ADP-ribosyl)transferase inhibitors. Such compounds are useful as therapeutics in treating cancers and in ameliorating the effects of stroke, head trauma, and neurodegenerative disease.
申请公布号 WO0116136(A3) 申请公布日期 2001.06.21
申请号 WO2000US23882 申请日期 2000.08.31
申请人 AGOURON PHARMACEUTICALS, INC.;CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED 发明人 WEBBER, STEPHEN, EVAN;SKALITZKY, DONALD, JAMES;TIKHE, JAYASHREE, GIRISH;KUMPF, ROBERT, ARNOLD;MARAKOVITS, JOSEPH, TIMOTHY;EASTMAN, WALTER, BRIAN
分类号 C07D487/04;A61K31/5517;A61P3/10;A61P5/50;A61P9/00;A61P9/10;A61P17/00;A61P25/00;A61P29/00;A61P35/00;A61P43/00;C07D487/06 主分类号 C07D487/04
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