发明名称 |
METHOD OF SYNTHESISING INHIBITORS OF HIV PROTEASE |
摘要 |
<p>An improved process for the synthesis of (3S)-tetrahydro-3-furyl N-[(1S,2R)-3 -(4-amino-N-isobutylbenzenesulphonamido)-1-benzyl-2-hydroxypropyl]carbamate comprising four steps form the compound of formula A and a novel intermediate thereto.</p> |
申请公布号 |
PL342602(A1) |
申请公布日期 |
2001.06.18 |
申请号 |
PL19990342602 |
申请日期 |
1999.03.18 |
申请人 |
GLAXO GROUP LTD |
发明人 |
AL-FARHAN EMILE;DEININGER DAVID D.;MCGHIE STEPHEN;O'CALLAGHAN JOHN;ROBERTSON MARK STUART;RODGERS KEITH;ROUT STEPHEN JOHN;SINGH HARDEV;TUNG ROGER DENNIS |
分类号 |
A61P31/18;C07C311/18;C07D307/20;(IPC1-7):C07D307/20;C07C311/17 |
主分类号 |
A61P31/18 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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