发明名称 METHOD OF PRODUCING KETONE DERIVATIVE AND SYNTHETIC INTERMEDIATE THEREFOR
摘要 PROBLEM TO BE SOLVED: To provide a new synthetic intermediate for a ketone derivative and a method for producing the new intermediate. SOLUTION: The objective new compound that is useful as a synthetic intermediate of a ketone derivative is represented by formula (II) (wherein R2 is H, an alkyl or the like; Q is an alkoxy-alkyl, tetrahydropyranyl or the like; L is an alkoxy, imidazol-1-yl or N-methyl-N-methoxyamino; n is 0, 1 or 2). The compound of formula (I) [wherein individual signals are synonymous with those in the formula (II)] is produced by allowing the new intermediate compound of formula (II) to react with a compound of formula (III): R1-M (wherein R1 is phenyl or a heterocyclic group or the like; M is a lithium or magnesium halide).
申请公布号 JP2001158761(A) 申请公布日期 2001.06.12
申请号 JP19990339734 申请日期 1999.11.30
申请人 SHIONOGI & CO LTD 发明人 KAI HIROYUKI;NAKAI TORU
分类号 C07D233/58;C07C45/45;C07C67/343;C07C69/78;C07C259/10;C07D307/20;C07D309/12;C07D335/02;C07D401/12;C07D405/12;C07D409/12;(IPC1-7):C07C69/78 主分类号 C07D233/58
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