发明名称 PARTIAL OR FULL A1 AGONISTS - N<6> HETEROCYCLIC 5'-THIO SUBSTITUTED ADENOSINE DERIVATIVES
摘要 N<6> heterocyclic 5' modified adenosine derivatives that are adenosine A1 receptor partial or full agonists, and as such, are useful for modifying cardiac activity, modifying adipocyte function, treating central nervous system disorders, and treating diabetic disorders and obesity in mammals, and especially in humans.
申请公布号 WO0140246(A1) 申请公布日期 2001.06.07
申请号 WO2000US32721 申请日期 2000.12.01
申请人 CV THERAPEUTICS, INC.;ZABLOCKI, JEFF, A.;PALLE, VENKATA, P.;VARKHEDKAR, VAIBHAV;BELARDINELLI, LUIZ 发明人 ZABLOCKI, JEFF, A.;PALLE, VENKATA, P.;VARKHEDKAR, VAIBHAV;BELARDINELLI, LUIZ
分类号 C07H19/167;A61K9/08;A61K9/20;A61K31/7076;A61P3/04;A61P3/10;A61P9/00;A61P9/04;A61P9/10;A61P25/00;A61P25/08;A61P43/00;C07H19/16;(IPC1-7):C07H19/16;A61K31/707 主分类号 C07H19/167
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