发明名称 HYDROXYETHOXYBENZAMIDE DERIVATIVES AND DRUGS CONTAINING THE SAME
摘要 Hydroxyethoxybenzamide derivatives represented by general formula (I), which have a dopamine D2 receptor blocking effect and a 5-HT4 receptor stimulating effect and are useful as drugs ameliorating digestive tract functions with the regulated expression of extrapyramidal syndrome, or pharmacologically acceptable salts thereof; wherein R<1> represents halogeno; R<2> represents hydrogen or halogeno; R<3> represents halogeno; and R<4> represents lower alkyl, lower alkoxy, amino, halo(lower alkyl) or halo(lower alkoxy). These compounds are efficacious for diseases such as reflux esophagitis, epigastric unidentified complaint, gastritis and gastric ulcer.
申请公布号 WO0136385(A1) 申请公布日期 2001.05.25
申请号 WO2000JP07790 申请日期 2000.11.07
申请人 KISSEI PHARMACEUTICAL CO., LTD.;OKAZAKI, KOSUKE;KOBAYASHI, HIROAKI;HORA, MASACHIYO;MASUDA, NAOYUKI;KITAZAWA, MAKIO 发明人 OKAZAKI, KOSUKE;KOBAYASHI, HIROAKI;HORA, MASACHIYO;MASUDA, NAOYUKI;KITAZAWA, MAKIO
分类号 A61P1/04;A61P1/08;A61P1/14;A61P43/00;C07D211/58;(IPC1-7):C07D211/58;A61K31/445 主分类号 A61P1/04
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