发明名称 |
2-benzyl and 2-heteroaryl benzimidazole nmda/nr2b antagonists |
摘要 |
Benzimidazoles, substituted in the 2-position by substituted benzyl groups or heteroaryl groups are effective as NMDA NR2B antagonists and are useful for relieving pain. |
申请公布号 |
AU1345001(A) |
申请公布日期 |
2001.05.14 |
申请号 |
AU20010013450 |
申请日期 |
2000.10.26 |
申请人 |
MERCK AND CO., INC. |
发明人 |
JOHN A. MCCAULEY;CORY R. THEBERGE;NIGEL J. LIVERTON;DAVID A. CLAREMON;CHRISTOPHER F. CLAIBORNE |
分类号 |
A61K31/4184;A61K31/4439;A61P25/04;A61P25/16;A61P25/18;A61P25/24;A61P43/00;C07D235/12;C07D401/06;C07D403/12;C07D405/12;C07D409/12;C07D413/12 |
主分类号 |
A61K31/4184 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|