发明名称 Sulphonyl compounds for use as linkers in solid phase and combinatorial synthesis
摘要 The present invention relates to a linker shown by the following formula (I):wherein R1 is a group of the formula (A):[wherein R3, R4 and R5 are the same or different hydrogen, etc], etc,R2 is a group which can form a chemical bond to a resin which may be protected by a conventional protective group,A is lower alkylene, etc,X is a leaving group, andm is an integer of 0 or 1,with proviso that A is (C2-C6)alkylene, andm is an integer of 1,when R1 is a group of the formula (A).
申请公布号 US6225480(B1) 申请公布日期 2001.05.01
申请号 US19990331580 申请日期 1999.06.30
申请人 FUJISAWA PHARMACEUTICAL CO., LTD. 发明人 TANAKA AKITO;TSUTSUMI HIDEO
分类号 C07B61/00;C07C309/87;C07C311/54;C07D311/70;C07D311/92;(IPC1-7):C07D311/04 主分类号 C07B61/00
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