| 发明名称 |
METHOD FOR PREPARING OXYCODONE |
| 摘要 |
A method for the preparation of oxycodone, and salts thereof, from codeine comprising oxidation of codeine to codeinone, formation of an dienolsilyl ether congener of codeinone in strong amine base, oxidation of the dienolsil yl ether congener using peracetic acid, and hydrogenation of the resulting 14- hydroxycodeinone product.
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| 申请公布号 |
CA2387523(A1) |
申请公布日期 |
2001.04.26 |
| 申请号 |
CA20002387523 |
申请日期 |
2000.09.15 |
| 申请人 |
BOEHRINGER INGELHEIM CHEMICALS, INC. |
发明人 |
LO, YOUNG S.;CHIU, FANG-TING |
| 分类号 |
C07D489/08;C07B61/00;C07D489/06;(IPC1-7):C07D489/02;A61P25/04;A61K31/485 |
主分类号 |
C07D489/08 |
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