摘要 |
PROBLEM TO BE SOLVED: To provide a method for producing N-acetylhomopiperazines in high yield by selectively acetylating one of amino groups in homopiperazines. SOLUTION: N-acetylhomopiperazines such as N-acetyl-1,4-diazacycloheptane and the like which are useful as intermediates for medicines are obtained by reacting homopiperazines with an acetylating agent in the presence of oxygen.
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