| 发明名称 |
1-PIPERAZINYL-2-BUTENES AND 2-BUTYNES, INTERMEDIATES THEREOF, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS |
| 摘要 |
HOE 91/S 002 The present invention relates to 1-piperazinyl-2-butenes and 2-butynes of the formula 1 <IMG> 1 wherein B is -C ? C-, <IMG> or <IMG> The invention relates furthermore to intermediates and a process for the preparation of the above compounds. The compounds of the formula 1 have antipsychotic activity and can, therefore, be used as medicaments.
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| 申请公布号 |
CA2059110(A1) |
申请公布日期 |
1992.07.11 |
| 申请号 |
CA19922059110 |
申请日期 |
1992.01.09 |
| 申请人 |
HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED |
发明人 |
ONG, HELEN H.;HRIB, NICHOLAS J.;PEREZ, JOSEPH;JURCAK, JOHN G. |
| 分类号 |
A61K31/495;A61P25/18;C07D209/48;C07D221/20;C07D239/42;C07D277/14;C07D277/20;C07D277/34;C07D295/12;C07D295/125;C07D401/12;C07D403/12;C07D409/00;C07D409/12;C07D417/12;C07D471/04;(IPC1-7):C07D403/06;C07D417/04;C07D401/06;C07D401/14;C07D403/14;C07D409/14;C07D417/14 |
主分类号 |
A61K31/495 |
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