发明名称 HETEROSUBSTITUTED PYRIDINE DERIVATIVES AS <i>PDE 4</i> INHIBITORS
摘要 The invention encompasses the novel compound of Formula (I) useful in the treatment of diseases, including asthma, by raising the level of cyclic adenosine-3',5'-monophosphate (cAMP) through the inhibition of phosphodiesterase IV (PDE 4) or a pharmaceutically acceptable salt or hydrate thereof. The invention also encompasses pharmaceutical compositions and methods for treatment.
申请公布号 WO0068198(A3) 申请公布日期 2001.04.05
申请号 WO2000CA00500 申请日期 2000.05.03
申请人 MERCK FROSST CANADA & CO.;COTE, BERNARD;FRIESEN, RICHARD;FRENETTE, RICHARD;GIRARD, MARIO;GIRARD, YVES;GODBOUT, CEDRICKX;GUAY, DANIEL;HAMEL, PIERRE;BLOUIN, MARC;DUCHARME, YVES;PRESCOTT, SYLVIE 发明人 COTE, BERNARD;FRIESEN, RICHARD;FRENETTE, RICHARD;GIRARD, MARIO;GIRARD, YVES;GODBOUT, CEDRICKX;GUAY, DANIEL;HAMEL, PIERRE;BLOUIN, MARC;DUCHARME, YVES;PRESCOTT, SYLVIE
分类号 A61K31/444;A61K31/4725;A61P1/04;A61P9/00;A61P9/10;A61P11/00;A61P11/06;A61P13/00;A61P13/12;A61P17/00;A61P17/06;A61P19/02;A61P25/00;A61P25/02;A61P25/24;A61P25/28;A61P27/02;A61P29/00;A61P31/00;A61P31/04;A61P31/10;A61P31/12;A61P35/00;A61P37/00;A61P37/06;A61P43/00;C07D213/74;C07D213/76;C07D213/79;C07D213/89;C07D401/14;C07D405/14;C07D409/14;C07D417/14;(IPC1-7):C07D213/89;A61K31/442 主分类号 A61K31/444
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