发明名称 |
Methods for the acylation of amine compounds |
摘要 |
Method for the acylation of amines are disclosed in which includes reacting a first reactant containing an amine group with a second reactant containing an acyl halide group, wherein the reaction takes place in the presence of secondary carboxylic acid salt form, of formula I:whereinR4 is an alkyl group having 1 to 10 carbon atoms; andR5 is an alkyl group having 1 to 10 carbon atoms.
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申请公布号 |
US6211384(B1) |
申请公布日期 |
2001.04.03 |
申请号 |
US19990385722 |
申请日期 |
1999.08.30 |
申请人 |
NOVARTIS PHARMACEUTICALS CORP. |
发明人 |
FITT, SR. JOHN JOSEPH;KAPA PRASAD KOTESWARA |
分类号 |
C07C231/02;C07D207/16;(IPC1-7):C07D207/04 |
主分类号 |
C07C231/02 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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