发明名称 PROCESSES FOR THE PREPARATION OF 4(5)-AMINO-5(4)-CARBOXAMIDOIMIDAZOLES AND INTERMEDIATES THEREOF
摘要 <p>The invention provides novel processes for preparing efficiently compounds of general formula (I) (wherein R1 and R2 are each independently hydrogen, optionally substituted C1-C10 alkyl, C3-C14 hydrocarbyl bearing an alicyclic skeleton, or the like) and intermediates thereof. Compounds of general formula (I) can be prepared by subjecting compounds of general formula (II) and/or salts thereof to cyclization hydrolysis in an aqueous basic solution. Further, compounds of general formula (II) can be prepared from industrially easily available diaminomaleonitrile in a high yield.</p>
申请公布号 WO2001021592(P1) 申请公布日期 2001.03.29
申请号 JP2000006397 申请日期 2000.09.20
申请人 发明人
分类号 主分类号
代理机构 代理人
主权项
地址