发明名称 |
ACETYLCHOLINE ENHANCERS |
摘要 |
Disclosed herein are quinoline derivatives having dual mechanistic properties, referred to in this patent document as "acetylcholine enhancers", i.e., compounds which evidence acetylcholinesterase (AChE) inhibition activity, and 5-HT3 receptor antagonist activity. A particularly preferred compound is 2-[2-(1-benzylpiperizin-4-yl) ethyl]-2,3-dihydro-9-methoxy-1H-pyrrolo [3,4-b] quinolin-1-one hemifumarate, referred to herein as Compound A ("Cm.A"). |
申请公布号 |
EP1086102(A1) |
申请公布日期 |
2001.03.28 |
申请号 |
EP19990933508 |
申请日期 |
1999.06.09 |
申请人 |
ARENA PHARMACEUTICALS, INC.;SSP CO., LTD. |
发明人 |
CHALMERS, DEREK, T.;SATO, SUSUMO;KODA, TADAYUKI |
分类号 |
A61K31/44;A61K31/4545;A61P25/28;A61P43/00;C07D471/04 |
主分类号 |
A61K31/44 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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