发明名称 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES
摘要 Disclosed are novel cathepsin S, K, F, L and B reversible inhibitory compounds of formulas (I), (II), (Ia) and (Ib) further defined herein. The compounds are useful for treating autoimmune diseases. Also disclosed are processes for making such novel compounds.
申请公布号 WO0119816(A1) 申请公布日期 2001.03.22
申请号 WO2000US23584 申请日期 2000.08.28
申请人 BOEHRINGER INGELHEIM PHARMACEUTICALS, INC.;EMMANUEL, MICHEL, J.;FRYE, LEAH, L.;HICKEY, EUGENE, R.;LIU, WEIMIN;MORWICK, TINA, M.;SPERO, DENICE, M.;SUN, SANXING;THOMSON, DAVID, S.;WARD, YANCEY, D.;YOUNG, ERICK, R., R. 发明人 EMMANUEL, MICHEL, J.;FRYE, LEAH, L.;HICKEY, EUGENE, R.;LIU, WEIMIN;MORWICK, TINA, M.;SPERO, DENICE, M.;SUN, SANXING;THOMSON, DAVID, S.;WARD, YANCEY, D.;YOUNG, ERICK, R., R.
分类号 A61K31/428;A61K31/4468;A61K31/4535;A61K31/454;A61K31/496;A61K31/4965;A61K31/506;A61K31/536;A61K31/5375;A61P1/04;A61P3/10;A61P5/14;A61P9/10;A61P11/06;A61P13/12;A61P17/00;A61P17/06;A61P19/08;A61P19/10;A61P21/04;A61P25/00;A61P25/02;A61P25/28;A61P29/00;A61P37/00;A61P37/02;A61P37/08;C07D205/04;C07D207/14;C07D207/16;C07D211/58;C07D211/66;C07D309/14;C07D335/02;C07D401/04;C07D401/12;C07D403/06;C07D409/12;C07D413/12;C07D417/12;C07D451/04;(IPC1-7):C07D401/12;A61K31/453 主分类号 A61K31/428
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