发明名称 2-`3-AMINO-4-(N-HYDROXYAMINO)-SUCCINYLAMINO-ACETAMIDES FOR USE AS CD23 FORMATION INHIBITORS
摘要 Compounds of formula (I): wherein X<1> is alkyl, sulphonyl or carboxy; X<2> is hydrogen or alkyl; R<1> is arylmethyl or heterocyclylmethyl; R<2> is alkyl, alkenyl, aryl, cycloalkyl or cycloalkenyl; and R<3> is hydrogen, alkyl, alkenyl, alkynyl or aryl; are useful in the treatment of disorders mediated by s-CD23.
申请公布号 WO0149657(A8) 申请公布日期 2001.11.08
申请号 WO2000GB05012 申请日期 2000.12.22
申请人 SMITHKLINE BEECHAM, PLC;FALLER, ANDREW;ROUSSEAU, ANNE-GERALDINE;MACPHERSON, DAVID, TIMOTHY;MILNER, PETER, HENRY 发明人 FALLER, ANDREW;ROUSSEAU, ANNE-GERALDINE;MACPHERSON, DAVID, TIMOTHY;MILNER, PETER, HENRY
分类号 A61P29/00;A61K31/16;A61K31/165;A61K31/18;A61P37/02;A61P37/08;A61P43/00;C07C259/06;C07C303/38;C07C311/13;C07D307/52;(IPC1-7):C07C259/06;A61K37/00 主分类号 A61P29/00
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