发明名称 Process for production of piperidine derivatives
摘要 The present invention relates to a method for preparing piperidine derivative compounds by converting, with a piperidine compound, regioisomers having the formula:and where m is an integer from 1 to 6; Q and Y are the same or different and are selected from the group consisting of O, S, and NR5; G1, G2, and G3 are the same or different and are selected from the group consisting of OR8, SR8, and NR8R9; R6 and R7 are the same or different and are selected from the group consisting of hydrogen, an alkyl moiety, an aryl moiety, OR8, SR8, and NR8R9; X3 is halogen, OR15, SR15, NR15R16, OSO2R15, or NHSO2R15; R5, R8, R9, R15, and R16 are the same or different and are selected from the group consisting of hydrogen, an alkyl moiety, and an aryl moiety; and A is a substituent of its ring and is selected from the group consisting of hydrogen, halogens, alkyl, hydroxy, alkoxy, and other substituents.
申请公布号 US6201124(B1) 申请公布日期 2001.03.13
申请号 US19950575344 申请日期 1995.12.21
申请人 ALBANY MOLECULAR RESEARCH, INC. 发明人 D'AMBRA THOMAS E.;PILLING GARRY M.
分类号 A61K31/00;A61K31/42;A61K31/421;A61K31/445;A61P37/00;A61P37/08;C07D211/22;C07D211/54;C07D261/04;C07D263/10;(IPC1-7):C07D211/34 主分类号 A61K31/00
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