发明名称 ANDROGEN RECEPTOR MODULATOR COMPOUNDS AND METHODS
摘要 Compounds, pharmaceutical compositions, and methods for modulating processes mediated by steroid receptors. In particular, preparation and methods of use of non-steroidal compounds and compositions that are agonists, partial agonists, and antagonists for the androgen receptor (AR) are described. Further, described are the methods of making and use of critical intermediates including a stereoselective synthetic route to intermediates for the AR modulators.
申请公布号 WO0116139(A1) 申请公布日期 2001.03.08
申请号 WO2000US23520 申请日期 2000.08.25
申请人 LIGAND PHARMACEUTICALS INCORPORATED;HIGUCHI, ROBERT;ARIENTI, KRISTEN, L.;NEELAKANDHA, MANI;PIO, BARBARA;ZHI, LIN;CHEN, PENGHUI;CAFERRO, THOMAS, R. 发明人 HIGUCHI, ROBERT;ARIENTI, KRISTEN, L.;NEELAKANDHA, MANI;PIO, BARBARA;ZHI, LIN;CHEN, PENGHUI;CAFERRO, THOMAS, R.
分类号 A61K31/4985;A61K31/5383;A61K31/542;A61P5/00;A61P5/24;A61P5/26;A61P5/28;A61P7/00;A61P7/06;A61P13/08;A61P15/08;A61P15/10;A61P15/16;A61P17/10;A61P17/14;A61P19/10;A61P35/00;C07D471/04;C07D498/04;C07D498/14;C07D513/04 主分类号 A61K31/4985
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