| 发明名称 |
METHOD OF SYNTHESIS OF PYRROLE AMIDES |
| 摘要 |
<p>A method for preparing pyrrole-carboxyamides with selectively bind to GABAa receptors, which comprises reacting 1,3-cycloakane-diones with bromoethylacetate followed by reaction of the resulting product with an acid halide followed by reaction with an aromatic amine and finally with an ammonium sources at an elevated temperature. 12 claims</p> |
| 申请公布号 |
BG104413(A) |
申请公布日期 |
2001.02.28 |
| 申请号 |
BG20000104413D |
申请日期 |
2000.05.09 |
| 申请人 |
PFIZER PRODUCTS INC |
发明人 |
RAGAN, JOHN A.;MAKOWSKI, TERESA W.;AM ENDE, DAVID J.;CLIFFORD, PAMELA J.;YOUNG, GREGORY R.;CONRAD, ALYSON K.;EISENBEIS, SHANE A.;QUALLICH, GEORGE J.;MELDRUM ALLEN, DOUGLAS JOHN |
| 分类号 |
C07D307/93;C07C271/14;C07D209/42;C07D209/52;C07D307/83;C07D307/84;C07D401/12;C07D405/12;C07D407/12;(IPC1-7):C07D209/42;A61K31/343;A61K31/403;A61P25/24 |
主分类号 |
C07D307/93 |
| 代理机构 |
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