发明名称 Substituted pyrazoles as p38 Kinase inhibitors.
摘要 A class of pyrazole derivatives is described for use in treating p38 kinase mediated disorders. Compounds of particular interest are defined by Formula (I) wherein R 1, R 2, R 3 and R 4 are as described in the specification.
申请公布号 KR20010012854(A) 申请公布日期 2001.02.26
申请号 KR19997010820 申请日期 1998.05.22
申请人 SEARLE & CO 发明人 ANANTANARAYAN ASHOK;CLARE MICHAEL;COLLINS PAUL W;CRICH JOYCE ZUOWU;DEVRAJ RAJESH;FLYNN DANIEL L;GENG LIFENG;HANSON GUNNAR J;KOSZYK FRANCIS J;LIAO SHUYUAN;PARTIS RICHARD A;RAO SHASHIDHAR N;SELNESS SHAUN RAJ;SOUTH MICHAEL J;STEALEY MICHAEL A;WEIER RICHARD M;XU XIANGDONG
分类号 C07D473/00;A61K31/4155;A61K31/422;A61K31/427;A61K31/4439;A61K31/454;A61K31/4545;A61K31/496;A61K31/498;A61K31/506;A61K31/52;A61K31/5377;A61P1/04;A61P3/14;A61P7/02;A61P9/10;A61P11/00;A61P11/06;A61P17/06;A61P19/02;A61P19/06;A61P29/00;A61P37/06;A61P43/00;C07D401/04;C07D401/14;C07D403/04;C07D405/14;C07D409/04;C07D409/14;C07D413/04;C07D413/14;C07D417/04;C07D417/14;C07D451/02;C07D453/02;C07D471/04;(IPC1-7):A47G19/22 主分类号 C07D473/00
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