发明名称 |
Substituted pyrazoles as p38 Kinase inhibitors. |
摘要 |
A class of pyrazole derivatives is described for use in treating p38 kinase mediated disorders. Compounds of particular interest are defined by Formula (I) wherein R 1, R 2, R 3 and R 4 are as described in the specification.
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申请公布号 |
KR20010012854(A) |
申请公布日期 |
2001.02.26 |
申请号 |
KR19997010820 |
申请日期 |
1998.05.22 |
申请人 |
SEARLE & CO |
发明人 |
ANANTANARAYAN ASHOK;CLARE MICHAEL;COLLINS PAUL W;CRICH JOYCE ZUOWU;DEVRAJ RAJESH;FLYNN DANIEL L;GENG LIFENG;HANSON GUNNAR J;KOSZYK FRANCIS J;LIAO SHUYUAN;PARTIS RICHARD A;RAO SHASHIDHAR N;SELNESS SHAUN RAJ;SOUTH MICHAEL J;STEALEY MICHAEL A;WEIER RICHARD M;XU XIANGDONG |
分类号 |
C07D473/00;A61K31/4155;A61K31/422;A61K31/427;A61K31/4439;A61K31/454;A61K31/4545;A61K31/496;A61K31/498;A61K31/506;A61K31/52;A61K31/5377;A61P1/04;A61P3/14;A61P7/02;A61P9/10;A61P11/00;A61P11/06;A61P17/06;A61P19/02;A61P19/06;A61P29/00;A61P37/06;A61P43/00;C07D401/04;C07D401/14;C07D403/04;C07D405/14;C07D409/04;C07D409/14;C07D413/04;C07D413/14;C07D417/04;C07D417/14;C07D451/02;C07D453/02;C07D471/04;(IPC1-7):A47G19/22 |
主分类号 |
C07D473/00 |
代理机构 |
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