发明名称 SUSTAINED RELEASE FORMULATION OF A PEPTIDE
摘要 This invention pertains to a sustained release complex, Compound (I), which comprises Compound (A), having formula (A) or a pharmaceutically acceptable salt thereof, and a copolymer comprising poly-(I)-lactic-glycolic-tartaric acid (P(I)LGT), wherein the amino group of said Compound (A) is ionically bound to a carboxyl group of the P(I)LGT. The present invention further pertains to a process for making said sustained release complex. Further still, the present invention is directed to a pharmaceutical composition comprising said sustained release complex and a pharmaceutically acceptable carrier(s).
申请公布号 WO0112233(A2) 申请公布日期 2001.02.22
申请号 WO2000US22464 申请日期 2000.08.16
申请人 SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES S.A.S.;MOREAU, JACQUES-PIERRE 发明人 MOREAU, JACQUES-PIERRE
分类号 A61K9/16;A61K38/00;A61K47/48;A61P1/00;A61P3/10;A61P9/02;A61P9/12;A61P17/06;A61P19/08;A61P21/04;A61P25/00;A61P35/00;C07D241/04;C07K7/06;(IPC1-7):A61K47/48 主分类号 A61K9/16
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