发明名称 HETEROSUBSTITUTED PYRIDINE DERIVATIVES AS <i>PDE 4</i> INHIBITORS
摘要 The invention encompasses the novel compound of Formula (I) useful in the treatment of diseases, including asthma, by raising the level of cyclic adenosine-3',5'-monophosphate (cAMP) through the inhibition of phosphodiesterase IV (PDE 4). The invention also encompasses pharmaceutical compositions and methods for treatment.
申请公布号 WO0064874(A3) 申请公布日期 2001.02.15
申请号 WO2000CA00427 申请日期 2000.04.19
申请人 MERCK FROSST CANADA & CO.;FRENETTE, RICHARD;FRIESEN, RICHARD;GIRARD, MARIO;GIRARD, YVES;GODBOUT, CEDRICKX;GUAY, DANIEL;HAMEL, PIERRE;PERRIER, HELENE 发明人 FRENETTE, RICHARD;FRIESEN, RICHARD;GIRARD, MARIO;GIRARD, YVES;GODBOUT, CEDRICKX;GUAY, DANIEL;HAMEL, PIERRE;PERRIER, HELENE
分类号 A61K31/443;A61K31/4436;A61K31/4439;A61K31/444;A61P9/00;A61P9/10;A61P11/00;A61P11/06;A61P17/00;A61P17/06;A61P19/02;A61P29/00;A61P35/00;A61P43/00;C07D213/64;C07D213/76;C07D213/79;C07D213/89;C07D405/14;C07D409/14;C07D417/14;(IPC1-7):C07D213/89;A61K31/442 主分类号 A61K31/443
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